Title of Invention

CHEMICAL COMPOUNDS CONTAINING TOCOPHEROL AND AT LEAST ONE ADDITIONAL PHARMACEUTICAL ACTIVE SUBSTANCE

Abstract The invention relates to chemical compounds in the form of their racemates, enantiomers or diastereomers with general formula I in which R stands for the unchanged portion of a variable pharmaceutical active ingredient molecule, B stands for a spacer, and Toc with the formula and R', R" and R''' are equal to H or methyl stands for tocopherol and A stands for C=X, SOm, X or CH2, whereby X is equal to 0, S or NR1 (when n 1) or S or NR1 (when n = 0), and B means a grouping X-R2-Y with Y equal to C=X, SOm or C(XR3)R4, and n is equal to 0 to 6, preferably 0, 1, 2 or 3, and m stands for 1 or 2, whereby R1 stands for H, C1 to C10-alkyl, preferably C1 to C6-alkyl or aryl, Het or an aryl or Het radical that is bonded via a C1 to C6-spacer, preferably C1 to C3, and whereby R2 is selected from the group alkylene, arylene or Het spacers as well as combinations thereof, whereby the latter are linked to one another either directly or via radical A or via grouping X0-A-Xp, whereby o and p are equal to 0, 1 or 2, and the latter can be the same or different, and whereby R3 and R4 stand for H, C1 to C10-alkyl, preferably C1-C6-alkyl or aryl, Het or an aryl or Het radical that is bonded via a C1 to C6 spacer, preferably C1 to C3-spacers.
Full Text

Documents:

00392-kolnp-2005 abstract.pdf

00392-kolnp-2005 claims.pdf

00392-kolnp-2005 correspondence.pdf

00392-kolnp-2005 correspondence_1.1.pdf

00392-kolnp-2005 correspondence_1.2.pdf

00392-kolnp-2005 correspondence_1.3.pdf

00392-kolnp-2005 description(complete).pdf

00392-kolnp-2005 form-1.pdf

00392-kolnp-2005 form-18.pdf

00392-kolnp-2005 form-3.1.pdf

00392-kolnp-2005 form-3.pdf

00392-kolnp-2005 form-5.pdf

00392-kolnp-2005 g.p.a.pdf

00392-kolnp-2005 international publication.pdf

00392-kolnp-2005 international search authority report.pdf

00392-kolnp-2005 pct others.pdf

00392-kolnp-2005 priority document.pdf

392-kolnp-2005-granted-abstract.pdf

392-kolnp-2005-granted-assignment.pdf

392-kolnp-2005-granted-claims.pdf

392-kolnp-2005-granted-correspondence.pdf

392-kolnp-2005-granted-description (complete).pdf

392-kolnp-2005-granted-examination report.pdf

392-kolnp-2005-granted-form 1.pdf

392-kolnp-2005-granted-form 13.pdf

392-kolnp-2005-granted-form 18.pdf

392-kolnp-2005-granted-form 3.pdf

392-kolnp-2005-granted-form 5.pdf

392-kolnp-2005-granted-gpa.pdf

392-kolnp-2005-granted-letter patent.pdf

392-kolnp-2005-granted-reply to examination report.pdf

392-kolnp-2005-granted-specification.pdf


Patent Number 222157
Indian Patent Application Number 392/KOLNP/2005
PG Journal Number 30/2008
Publication Date 25-Jul-2008
Grant Date 23-Jul-2008
Date of Filing 10-Mar-2005
Name of Patentee JSW-RESEARCH FORSCHUNGSLABOR GMBH
Applicant Address RANKENGASSE 28, A-8020 GRAZ
Inventors:
# Inventor's Name Inventor's Address
1 WINDISCH MANFRED RANKENGASSE 28, A-8020 GRAZ
2 MATUSZCZAK BARBARA HERZOG-FRIEDRICH-STR,11, A-6020 INNSBRUCK
PCT International Classification Number C07D 405/12
PCT International Application Number PCT/AT2004/000234
PCT International Filing date 2004-07-01
PCT Conventions:
# PCT Application Number Date of Convention Priority Country
1 A 1127/2003 2003-07-17 Austria