Title of Invention

AN ORALLY ADMINISTERABLE GALENIC FORMULATION ALLOWING IMPROVED ABSORPTION BY THE TRANSMEMBRANE IN THE GASTROINTESTINAL TRACT.

Abstract The present invention relates to an orally administrable galenic form allowing improved absorption by the transmembrane or paracellular route in the gastrointestinal tract of active ingredients which are hydrophilic or ionizable in physiological media, comprising at least one such active ingredient, an absorption-promoting agent having an HLB greater than 8, the said absorption-promoting agent consisting of one or more lipid substances chosen from: polysorbates: ethers of polyoxyethylene and alkyl; esters of polyoxyethylene and fatty acids; fatty acids; fatty alcohols; bile acids and their salts with pharmaceutically acceptable cations; esters of C1-C6 alkanol with fatty acids, esters of polyol with fatty acids, the said polyol comprising from 2 to 6 hydroxyl functional groups; and polyglycolysed glycerides; in combination with one or more pharmaceutically acceptable excipients, the pharmaceutical forms comprising captopril being excluded.
Full Text

Documents:

IN-PCT-2000-233-KOL-(22-12-2011)-FORM-27.pdf

IN-PCT-2000-233-KOL-FORM-27.pdf

in-pct-2000-233-kol-granted-abstract.pdf

in-pct-2000-233-kol-granted-claims.pdf

in-pct-2000-233-kol-granted-correspondence.pdf

in-pct-2000-233-kol-granted-description (complete).pdf

in-pct-2000-233-kol-granted-drawings.pdf

in-pct-2000-233-kol-granted-examination report.pdf

in-pct-2000-233-kol-granted-form 1.pdf

in-pct-2000-233-kol-granted-form 18.pdf

in-pct-2000-233-kol-granted-form 2.pdf

in-pct-2000-233-kol-granted-form 26.pdf

in-pct-2000-233-kol-granted-form 3.pdf

in-pct-2000-233-kol-granted-form 5.pdf

in-pct-2000-233-kol-granted-letter patent.pdf

in-pct-2000-233-kol-granted-reply to examination report.pdf

in-pct-2000-233-kol-granted-specification.pdf

in-pct-2000-233-kol-granted-translated copy of priority document.pdf


Patent Number 219534
Indian Patent Application Number IN/PCT/2000/233/KOL
PG Journal Number 19/2008
Publication Date 09-May-2008
Grant Date 07-May-2008
Date of Filing 21-Aug-2000
Name of Patentee MERCK PATENT GMBH.
Applicant Address FRANKFURTER STRASSE 250, 64293 DARMSTADT
Inventors:
# Inventor's Name Inventor's Address
1 SASLAWSKI, OLIVIER 43 RUE DE SEZE 69006 LYON
2 GIET, PHILIPPE 9, PLACE TOBIE ROBATEL 69001 LYON
3 MICHEL, DOMINIQUE 284, RUE ANDRE PHILIP 69003 LYON
4 HULOT, THIERRY 24 RUE JARENTE 69002 LYON
PCT International Classification Number A 61 K 9/16
PCT International Application Number PCT/EP99/00994
PCT International Filing date 1999-02-16
PCT Conventions:
# PCT Application Number Date of Convention Priority Country
1 98/02143 1998-02-23 France