Title of Invention

INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1

Abstract The present invention discloses novel compounds of Formula I: ( I ) possessing 11β-HSD type 1 antagonist activity, as well as methods for preparing such compounds. In another embodiment, the invention discloses pharmaceutical compositions comprising compounds of Formula I, as well as methods of using the compounds and compositions to treat diabetes, hyperglycemia, obesity, hypertension, hyperlipidemia, metabolic syndrome, cognitive disorders, and other conditions associated with 11β-HSD type 1 activity.
Full Text PLEASE SEE THE SPECIFICATION ATTACHED.

Documents:

2277-mumnp-2008-abstract(23-10-2008).pdf

2277-MUMNP-2008-ASSIGNMENT(24-12-2008).pdf

2277-mumnp-2008-claims(23-10-2008).pdf

2277-MUMNP-2008-CLAIMS(AMENDED)-(15-5-2012).pdf

2277-mumnp-2008-claims(amended)-(4-11-2008).pdf

2277-MUMNP-2008-CLAIMS(GRANTED).pdf

2277-MUMNP-2008-CLAIMS(MARKED COPY)-(15-5-2012).pdf

2277-MUMNP-2008-CORRESPONDENCE(13-4-2009).pdf

2277-MUMNP-2008-CORRESPONDENCE(14-9-2011).pdf

2277-MUMNP-2008-CORRESPONDENCE(17-1-2013).pdf

2277-MUMNP-2008-CORRESPONDENCE(24-12-2008).pdf

2277-MUMNP-2008-CORRESPONDENCE(26-7-2012).pdf

2277-MUMNP-2008-CORRESPONDENCE(30-8-2012).pdf

2277-MUMNP-2008-CORRESPONDENCE(IPO).pdf

2277-mumnp-2008-description(complete)-(23-10-2008).pdf

2277-MUMNP-2008-DESCRIPTION(GRANTED).pdf

2277-MUMNP-2008-EP DOCUMENT(15-5-2012).pdf

2277-mumnp-2008-form 1(23-10-2008).pdf

2277-MUMNP-2008-FORM 1(30-8-2012).pdf

2277-MUMNP-2008-FORM 13(26-7-2012).pdf

2277-mumnp-2008-form 13(4-11-2008).pdf

2277-mumnp-2008-form 18(4-11-2008).pdf

2277-mumnp-2008-form 2(23-10-2008).pdf

2277-mumnp-2008-form 2(title page)-(23-10-2008).pdf

2277-MUMNP-2008-FORM 2(TITLE PAGE)-(GRANTED).pdf

2277-MUMNP-2008-FORM 26(14-9-2011).pdf

2277-MUMNP-2008-FORM 26(15-5-2012).pdf

2277-MUMNP-2008-FORM 3(13-4-2009).pdf

2277-MUMNP-2008-FORM 3(15-5-2012).pdf

2277-mumnp-2008-form 3(23-10-2008).pdf

2277-mumnp-2008-form 5(23-10-2008).pdf

2277-MUMNP-2008-FORM2(GRANTED).pdf

2277-mumnp-2008-marked copy(4-11-2008).pdf

2277-MUMNP-2008-PCT CLAIMS(15-5-2012).pdf

2277-MUMNP-2008-PETITION UNDER RULE 137(15-5-2012).pdf

2277-MUMNP-2008-PETITION UNDER RULE-137(17-1-2013).pdf

2277-MUMNP-2008-REPLY TO EXAMINATION REPORT(15-5-2012).pdf

2277-MUMNP-2008-US DOCUMENT(15-5-2012).pdf

2277-mumnp-2008-wo international publication report(23-10-2008).pdf

abstract1.jpg

Form-1.pdf

Form-3.pdf

Form-5.pdf


Patent Number 255425
Indian Patent Application Number 2277/MUMNP/2008
PG Journal Number 08/2013
Publication Date 22-Feb-2013
Grant Date 20-Feb-2013
Date of Filing 23-Oct-2008
Name of Patentee ELI LILLY AND COMPANY
Applicant Address LILLY CORPORATE CENTER, INDIANAPOLIS, INDIANA 46285,
Inventors:
# Inventor's Name Inventor's Address
1 LI, RENHUA 10493 Hollowood Court Fishers Indiana 46038 USA
2 WALLACE, OWEN, BRENDAN 13297 Mink Lane Westfield Indiana 46074 USA
3 XU, YANPING 6676 Pennan Court Noblesville Indiana 46062 USA
PCT International Classification Number C07D401/14
PCT International Application Number PCT/US2007/067353
PCT International Filing date 2007-04-25
PCT Conventions:
# PCT Application Number Date of Convention Priority Country
1 60/745,565 2006-04-25 U.S.A.