Title of Invention

NOVEL DIPEPTIDYL PEPTIDASE IV INHIBITORS, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Abstract The present invention relates to novel antidiabetic, hypolipidemic, and anticholesteromic, antiobesity compounds representated by formula I, where R,Rl,R2,R3,A,B,m,n are as defined ,their derivatives, their analogs, their tautomeric forms, their stereoisomers, their diastereomers , their bioisosteres, their polymorphs, their pharmaceutically acceptable salts and pharmaceutically acceptable compositions containing them. More specifically, the present invention relates to compounds of the general formula I which are predominantly serine protease inhibitors, particularly dipeptidyl peptidase inhibitors, more particularly dipeptidyl peptidase IV inhibitors, their derivatives, their analogs, their tautomeric forms, their stereoisomers, their diastereomers , their bioisosteres, their polymorphs, their pharmaceutically acceptable salts and pharmaceutically acceptable compositions containing them. The present invention also relates to the processes for the preparation of novel compounds of formula I and novel intermediates and also their use as antidiabetic, hypolipidemic, anticholesteromic and antiobesity compounds
Full Text

Documents:

610 -che-2006-abstarct.pdf

610 -che-2006-correspondance-others.pdf

610 -che-2006-correspondance-po.pdf

610 -che-2006-description provisional.pdf

610 -che-2006-form 1.pdf

610 -che-2006-form 3.pdf

610-CHE-2006 AMENDED CLAIMS 19-12-2011.pdf

610-CHE-2006 AMENDED CLAIMS 29-09-2011.pdf

610-CHE-2006 CORRESPONDENCE OTHERS 15-09-2011.pdf

610-CHE-2006 CORRESPONDENCE OTHERS 19-12-2011.pdf

610-CHE-2006 EXAMINATION REPORT REPLY RECEIVED 29-09-2011.pdf

610-CHE-2006 FORM-1 29-09-2011.pdf

610-CHE-2006 FORM-13 29-09-2011.pdf

610-CHE-2006 FORM-3 15-09-2011.pdf

610-CHE-2006 FORM-3 29-09-2011.pdf

610-CHE-2006 OTHER PATENT DOCUMENT 15-09-2011.pdf

610-CHE-2006 CLAIMS.pdf

610-CHE-2006 CORRESPONDENCE OTHERS 10-02-2012.pdf

610-CHE-2006 CORRESPONDENCE OTHERS 15-09-2011.pdf

610-CHE-2006 CORRESPONDENCE OTHERS 20-02-2012.pdf

610-CHE-2006 CORRESPONDENCE OTHERS.pdf

610-CHE-2006 CORRESPONDENCE PO.pdf

610-CHE-2006 CORRESPONDENCE. OTHERS 20-02-2012.pdf

610-che-2006 description (complete) 27-03-2007.pdf

610-CHE-2006 FORM-13 10-02-2012.pdf

610-CHE-2006 FORM-18.pdf

610-CHE-2006 FORM-3 15-09-2011.pdf

610-CHE-2006 FORM-3 16-07-2012.pdf

610-CHE-2006 POWER OF ATTORNEY.pdf

610-CHE-2006 CORRESPONDENCE-OTHERS 21-10-2009.pdf

610-che-2006 correspondene others 14-08-2007.pdf


Patent Number 251197
Indian Patent Application Number 610/CHE/2006
PG Journal Number 09/2012
Publication Date 02-Mar-2012
Grant Date 29-Feb-2012
Date of Filing 03-Apr-2006
Name of Patentee MATRIX LABORATORIES LTD.
Applicant Address 1-1-151/1, IV FLOOR, SAIRAM TOWERS, ALEXANDER ROAD SECUNDERABAD 500 003
Inventors:
# Inventor's Name Inventor's Address
1 DR. GOPALAN BALASUBRAMANIAN 1-1-151/1, IV FLOOR, SAIRAM TOWERS, ALEXANDER ROAD SECUNDERABAD 500 003
2 DR. RAVO DHAMJEWAR 1-1-151/1, IV FLOOR, SAIRAM TOWERS, ALEXANDER ROAD SECUNDERABAD 500 003
3 DR. RASHEED MOHAMMED 1-1-151/1, IV FLOOR, SAIRAM TOWERS, ALEXANDER ROAD SECUNDERABAD 500 003
4 DR. SREEDHARA SWAMYH KESHAVAPURA HOSAMANE 1-1-151/1, IV FLOOR, SAIRAM TOWERS, ALEXANDER ROAD SECUNDERABAD 500 003
PCT International Classification Number C07D401/12
PCT International Application Number N/A
PCT International Filing date
PCT Conventions:
# PCT Application Number Date of Convention Priority Country
1 NA