| Title of Invention | BENZENESULFONAMIDE DERIVATIVE OF FORMULA I |
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| Abstract | The present invention relates to a benzenesulfonamide derivative of formula (I), which is useful as an active ingredient of pharmaceutical preparations. The benzenesulfonamide derivatives of the present invention have CCR3 (CC type chemokine receptor) antagonistic activity, and can be used for the prophylaxis and treatment of diseases associated with CCR3 activity, in particular for the treatment of asthma, atopic dermatitis, allergic rhinitis and other inflammatory/immunological disorders. In said formula, X represents O or S; R4 represents formulae (a), (b), (c), (d), (e), (f), (g), (h), (i) or (j), the other substituents are as defined in claim 1. |
| Full Text | The present invention relates to a benzenesulfonamide derivative of formula (I), which is useful as an active ingredient of pharmaceutical preparations. The benzenesulfonamide derivatives of the present invention have CCR3 (CC type chemokine receptor) antagonistic activity, and can be used for the prophylaxis and treatment of diseases associated with CCR3 activity, in particular for the treatment of asthma, atopic dermatitis, allergic rhinitis and other inflammatory/immunological disorders. In said formula, X represents O or S; R4 represents formulae (a), (b), (c), (d), (e), (f), (g), (h), (i) or (j), the other substituents are as defined in claim 1. |
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2728-chenp-2005 complete specification as granted.pdf
2728-CHENP-2005 CORRESPONDENCE OTHERS.pdf
2728-CHENP-2005 CORRESPONDENCE PO.pdf
2728-CHENP-2005 DESCRIPTION (COMPLETE).pdf
2728-CHENP-2005 POWER OF ATTORNEY.pdf
| Patent Number | 235248 | ||||||||||||||||||||||||||||||||||||
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| Indian Patent Application Number | 2728/CHENP/2005 | ||||||||||||||||||||||||||||||||||||
| PG Journal Number | 29/2009 | ||||||||||||||||||||||||||||||||||||
| Publication Date | 17-Jul-2009 | ||||||||||||||||||||||||||||||||||||
| Grant Date | 29-Jun-2009 | ||||||||||||||||||||||||||||||||||||
| Date of Filing | 21-Oct-2005 | ||||||||||||||||||||||||||||||||||||
| Name of Patentee | ACTIMIS PHARMACEUTICALS, INC., | ||||||||||||||||||||||||||||||||||||
| Applicant Address | 11099 NORTH TORREY PINES ROAD, LA JOLLA, CA 92037 | ||||||||||||||||||||||||||||||||||||
Inventors:
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| PCT International Classification Number | A61K31/4965 | ||||||||||||||||||||||||||||||||||||
| PCT International Application Number | PCT/EP2004/002496 | ||||||||||||||||||||||||||||||||||||
| PCT International Filing date | 2004-03-11 | ||||||||||||||||||||||||||||||||||||
PCT Conventions:
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