| Title of Invention | A COMPOUND OF FORMULA 1 FOR INHIBITING THE ACTIVITY OF GPCR |
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| Abstract | A compound of formula I for inhibiting the activity of GPCR, said compound having the formula: wherein the ring may be of any configuration; Z is selected from the group consisting of: sulphur, oxygen, or NRA wherein RA is selected from the set defined for R1 to R5 or C1 to C15 acyl, C4 to C15 arylacyl or C4 to C15 heteroarylacyl, with the proviso that both R1 and RA are not hydrogen, X is selected from the group consisting of: oxygen or NRA providing that at least one X of General Formula I is NRA, R1 to R5 are independently selected from the group consisting of: H, C1 to C12 alkyl, C1 to C12 alkenyl, C1 to C12 alkynyl, C1 to C12 heteroalkyl, C4 to C15 aryl, C4 to C15 heteroaryl, C4 to C15 arylalkyl or C4 to C15 heteroarylalkyl substituent, wherein, when X is NRA, both RA and the corresponding R1 to R5 are not hydrogen. |
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858-kolnp-2005-granted-abstract.pdf
858-kolnp-2005-granted-claims.pdf
858-kolnp-2005-granted-correspondence.pdf
858-kolnp-2005-granted-description (complete).pdf
858-kolnp-2005-granted-examination report.pdf
858-kolnp-2005-granted-form 1.pdf
858-kolnp-2005-granted-form 13.pdf
858-kolnp-2005-granted-form 18.pdf
858-kolnp-2005-granted-form 2.pdf
858-kolnp-2005-granted-form 26.pdf
858-kolnp-2005-granted-form 3.pdf
858-kolnp-2005-granted-form 5.pdf
858-kolnp-2005-granted-letter patent.pdf
858-kolnp-2005-granted-reply to examination report.pdf
858-kolnp-2005-granted-specification.pdf
| Patent Number | 221016 | |||||||||||||||||||||
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| Indian Patent Application Number | 858/KOLNP/2005 | |||||||||||||||||||||
| PG Journal Number | 24/2008 | |||||||||||||||||||||
| Publication Date | 13-Jun-2008 | |||||||||||||||||||||
| Grant Date | 11-Jun-2008 | |||||||||||||||||||||
| Date of Filing | 11-May-2005 | |||||||||||||||||||||
| Name of Patentee | ALCHEMIA LIMITED | |||||||||||||||||||||
| Applicant Address | 3 HI-TECH COURT, BRISBANE TECHNOLOGY PARK, EIGHT MILES PLAINS, QUEENSLAND 4113 | |||||||||||||||||||||
Inventors:
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| PCT International Classification Number | A 61K 31/7008 | |||||||||||||||||||||
| PCT International Application Number | PCT/AU03/001347 | |||||||||||||||||||||
| PCT International Filing date | 2003-10-10 | |||||||||||||||||||||
PCT Conventions:
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