Title of Invention

AN AZULENE DERIVATIVE AND SALT THEREOF

Abstract THE PRESENT INVENTION PPROCVIDES AN AZULENE DERIVATIVE AND A SALT THJEREOFR, WHEREIN AN AZULEE RING IS BONDED TO A BEBZENE RING DIRECTLY OR VIA A LOWE ALKYLENE WHICH MAY NE SUBSTITUTED WITH A HALOGEN ATOM AND THE NENZENE RING IS DIRECTLY BONDED TO THE GLUCOSE RESIDUEM MAND IS IS USABLE AS A NA-GLUCOSE COTRANSPORTER INHIBNITOR, ESPECIALLY FOR A THEREPEUTIC AND /OR PREVENTIVE AGENT FOR DIABVTES SUCH AS INSULIN-DEPENDENT DIABETES (TYPE 1 DIABVETES AND INSULIN-INDEPENDENT DIABETES (TYPE 2 DIABETES), ASW WELL AS DIABETES-RELATED DISEASES SUCH AS ISULIN-RESISTANT DISEASES AND OBESITY.
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Documents:

1775-kolnp-2004-granted-abstract.pdf

1775-kolnp-2004-granted-claims.pdf

1775-kolnp-2004-granted-correspondence.pdf

1775-kolnp-2004-granted-description (complete).pdf

1775-kolnp-2004-granted-examination report.pdf

1775-kolnp-2004-granted-form 1.pdf

1775-kolnp-2004-granted-form 13.pdf

1775-kolnp-2004-granted-form 18.pdf

1775-kolnp-2004-granted-form 2.pdf

1775-kolnp-2004-granted-form 26.pdf

1775-kolnp-2004-granted-form 3.pdf

1775-kolnp-2004-granted-form 5.pdf

1775-kolnp-2004-granted-letter patent.pdf

1775-kolnp-2004-granted-reply to examination report.pdf

1775-kolnp-2004-granted-specification.pdf

1775-kolnp-2004-granted-translated copy of priority document.pdf


Patent Number 215535
Indian Patent Application Number 01775/KOLNP/2004
PG Journal Number 09/2008
Publication Date 29-Feb-2008
Grant Date 27-Feb-2008
Date of Filing 23-Nov-2004
Name of Patentee ASTELLAS PHARMA INC.. AND KOTOBUKI PHARMACEUTICAL CO. LTD.
Applicant Address 3-11, NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411` JAPAN; & 6351,OAZA-SAKAKI,SAKAKI MACHI, HANISHINA- GUN, NAGANO 389-0697, JAPAN
Inventors:
# Inventor's Name Inventor's Address
1 HIROSHI TOMITYAMA C/O KO5OBUKI P0HARMACEUTICAL CO.,LTD 6351,OAZA SAKAKI, SAKAKIMACHI HANISHINA GUM NAGANO 389-0697 JAPAN
2 ATSUSHI NODA 3--11, NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411` JAPAN
3 YOSHINORI KOBAYASHI 3--11, NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411` JAPAN
4 MASAKAZU IMAMURA C/O. YAMANOUCHI PHARMACEUTICAL CO.LTD., 21MIYUKIGAOKA TSUKUBASHIO IBARAKI 305-8585 JAPAN
5 TAKESHI KURAKAMI C/O YANMANOUDHI P0HARMACERUTICAL., LTSD 21 MIYUKIGAOKA, TSUKUBA SHI IBARAKI 305 8585, JAPAN
6 KAYOKA KITTA 3--11, NIHONBASHI-HONCHO 2-CHOME, CHUO-KU, TOKYO 103-8411` JAPAN
7 TAKAYUKI SUZUKI C/O YAMANOUCHI PHYARMACEUTICL CO., LTD 21, MIYUKIGAOKA, TSUKUBA SHI IBARKI 305-8585 JAPAN
8 EIJI KU8ROSAKI C/O YAMANOUCHI PAHARMACE7TIC AL CO9., LTD 21, MIYUKIGAOKA, TSUKUBA SHI IBARAKI 305-8585 JAPAN
PCT International Classification Number C07D309/12
PCT International Application Number PCT/JP03/009868
PCT International Filing date 2003-08-04
PCT Conventions:
# PCT Application Number Date of Convention Priority Country
1 2002-226869 2002-08-05 Japan
2 2003-130991 2003-05-09 Japan